Cascade bicyclization of triethylammonium thiolates with hydrazines: efficient access to pyrazolo[3,4-c]quinolines.

نویسندگان

  • Wei Fan
  • Yan-Rong Li
  • Bo Jiang
  • Guigen Li
چکیده

A new bicyclization strategy has been established, allowing a flexible and practical approach to 33 examples of pyrazolo[3,4-c]quinolines from low-cost and readily accessible triethylammonium thiolates with hydrazines. Notably, the features of this work include broad functional group compatibility, mild reaction conditions and good reaction yields.

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عنوان ژورنال:
  • Organic & biomolecular chemistry

دوره 14 38  شماره 

صفحات  -

تاریخ انتشار 2016